Publication

Original Paper (2020~present / 2016~2019 / before 2015)/Review, book, etc

Acylalkylation of Arynes Generated from o-Iodoaryl Triflates with Hydrosilanes and Cesium Fluoride

109

M. Minoshima, K. Uchida, Y. Nakamura, T. Hosoya,

*S. Yoshida

Diverse diaryl sulfide synthesis through consecutive aryne reactions

107

H. Nakajima, Y. Hazama, Y. Sakata, K. Uchida, T. Hosoya, *S. Yoshida

Chem. Commun. 2021, 57, 2621.

https://doi.org/10.1039/D0CC08373A

S1PR3–G12-biased agonist ALESIA targets cancer metabolism and promotes glucose starvation

108

M. Toyomoto, A. Inoue, K. Iida, M. Denawa, I. Kii, F. Marie, N. Kadji, T. Kishi, D. Im, T. Shimamura, H. Onogi, S. Yoshida, S. Iwata, J. Aoki, T. Hosoya, *M. Hagiwara

Cell Chem. Biol. 2021, in press.

https://doi.org/10.1016/j.chembiol.2021.01.004

Assembly of four modules onto a tetraazide platform by consecutive 1,2,3-triazole formations

106

*S. Yoshida, Y. Sakata, Y. Misawa, T. Morita, T. Kuribara, H. Ito, Y. Koike, I. Kii, *T. Hosoya

Chem. Commun. 2021, 57, 899.

https://doi.org/10.1039/D0CC07789E

Transition-Metal-Free Synthesis of N-Arylphenothiazines through an N- and S-Arylation Sequence

110

T. Matsuzawa, T. Hosoya, *S. Yoshida

Palladium-Catalyzed Sulfinylation of Aryl- and Alkenylborons with Sulfinate Esters

111

M. Suzuki, K. Kanemoto, Y. Nakamura, T. Hosoya,

*S. Yoshida

112

Nucleophilic transformations of azido-containing carbonyl compounds via protection of azido group

T. Aimi, T. Meguro, A. Kobayashi, *T. Hosoya, *S. Yoshida

Chem. Commun. 2021, 57, 6062.

https://doi.org/10.1039/D1CC01143J

113

Facile Synthetic Methods for Diverse N-Arylphenylalanine Derivatives via Transformations of Aryne Intermediates and Cross-Coupling Reactions

T. Kobayashi, T. Hosoya, *S. Yoshida

Bull. Chem. Soc. Jpn. 2021, 94, 1823.

https://doi.org/10.1246/bcsj.20210149

114

Thioxanthone Synthesis from Benzoic Acid Esters through Directed ortho-Lithiation

A. Kobayashi, T. Matsuzawa, T. Hosoya, *S. Yoshida

Chem. Lett. 2021, 50, 1624. [Selected as Editor's Choice (優秀論文)]

https://doi.org/10.1246/cl.210293

115

Synthesis of Azidoanilines by the Buchwald–Hartwig Amination

Y. Sakata, S. Yoshida, *T. Hosoya

J. Org. Chem. 2021, 86, 15674.

https://doi.org/10.1021/acs.joc.1c02251

116

Multicomponent click assembly through 2-azidoacrylamides

having a nucleophilic amino group


H. Takemura, G. Orimoto, A. Kobayashi, T. Hosoya,

S. Yoshida*

Org. Biomol. Chem. 2022, 20, 6007.

[New Talent 2022 themed issue]

https://doi.org/10.1039/D2OB00151A

117

Hydride reduction of o-(fluorosilyl)benzodifluorides for subsequent C–F transformations

R. Idogawa, A. Kobayashi, Y. Kim, K. Shimomori, T. Hosoya, S. Yoshida*

Chem. Commun. 2022, 58, 3521.

https://doi.org/10.1039/D1CC06761C

118

Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes


A. Nagai, A. Kobayashi, Y. Sakata, Y. Minami,

K. Uchida, T. Hosoya, S. Yoshida*

Synthesis 2022, 54, 5017.

[Special topic: Aryne Chemistry in Synthesis]

https://doi.org/10.1055/a-1834-2927

120

Pyridazine Synthesis from 1,2,4,5-Tetrazines and Alkynes in 1,1,1,3,3,3-Hexafluoro-2-propanol through the Inverse Electron Demand Diels–Alder Reaction

C. Yamamoto, M. Suzuki, S. Yoshida*

Bull. Chem. Soc. Jpn. 2022, 95, 1741. [BCSJ award article]

https://doi.org/10.1246/bcsj.20220267

119

Azido-type-selective triazole formation by iridium-catalyzed cycloaddition with thioalkynes


K. Sugiyama, Y. Sakata, T. Niwa, S. Yoshida, *T. Hosoya

Chem. Commun. 2022, 58, 6235.

https://doi.org/10.1039/D2CC01739C

121

Synthesis of benzo[b]furans from alkynyl sulfoxides and phenols by the interrupted Pummerer reaction

A. Kobayashi, T. Matsuzawa, T. Hosoya, S. Yoshida*

RSC Adv. 2023, 13, 839.

https://doi.org/10.1039/D2RA07856B

122

Migrative Thioamination of Aryne Intermediates Generated from o-Iodoaryl Triflates

S. Tabata, M. Minoshima, A. Kobayashi, T. Hosoya, S. Yoshida*

Synlett 2023, in press.

https://doi.org/10.1055/s-00000083


123

Fluorenones and Xanthones through Intramolecular C–F Arylation.

S. Hamada, S. Yoshida*

Bull. Chem. Soc. Jpn. 2023, in press.

https://doi.org/10.1246/bcsj.20230042

129

Bromothiolation of Arynes for the Synthesis of 2-Bromobenzenethiol Equivalents

S. Tabata, *S. Yoshida

130

Iterative click reactions using trivalent platforms for sequential molecular assembly

G. Orimoto, *S. Yoshida

Chem. Commun. 2024, 60, 5824.

https://doi.org/10.1039/D4CC01177E

131

Click assembly through selective azaylide formation

M. Hamada, G. Orimoto, *S. Yoshida

Chem. Commun. 2024, 60, 7930.

https://doi.org/10.1039/D4CC02723J

132

Regioselective pyridazine synthesis from tetrazines and alkynyl sulfides

C. Yamamoto, K. Numata, M. Suzuki, *S. Yoshida

Org. Chem. Front. 2024, 11, 6159.

https://doi.org/10.1039/D4QO01286K

133

Synthesis of Thiaphenanthridinones from Sulfinate Esters and 2-Borylanilines

K. Nakamura, M. Suzuki, S. Yoshida*

135

Thioxanthone Synthesis from Thioureas through Double Aryne Insertion into a Carbon–Sulfur Double Bond

M. Kawada, S. Tabata, Y. Hoshi, S. Yoshida*

134

Three-step click assembly using trivalent platforms bearing azido, ethynyl, and fluorosulfonyl groups


T. Yasuda, G. Orimoto, *S. Yoshida

Chem. Commun. 2025, 61, 2333.

https://doi.org/10.1039/d4cc06585a

136

Synthesis of multisubstituted naphthalenes through consecutive aryne reactions

T. Tanaka, S. Tabata, K. Nakamura, Y. Hazama, Y. Sakata, T. Hosoya, S. Yoshida*

Bull. Chem. Soc. Jpn. 2025, 98, uoaf001. [Selected paper, highlighted in Synfacts]

https://doi.org/10.1093/bulcsj/uoaf001

137

Synthesis of α-arylacetophenone derivatives by Grignard reactions and transformations of arynes via C–C bond cleavage

Y. Hoshi, S. Tabata, S. Yoshida*

Chem. Commun. 2025, 61, 3752.

https://doi.org/10.1039/D4CC06769J


138

Conditional fluorescent changes of azaylides with fluorescent chromophores

M. Hamada, S. Yoshida*

Chem. Lett. 2025, 54, upaf033.

https://doi.org/10.1093/chemle/upaf033

127

Facile synthesis of dibenzothiophene S-oxides from sulfinate esters

Y. Kumagai, A. Kobayashi, K. Nakamura, *S. Yoshida

Chem. Commun. 2024, 60, 1611.

https://doi.org/10.1039/D3CC05703H

128

Highly substituted benzo[b]furan synthesis through substituent migration

A. Kobayashi, S. Tabata, *S. Yoshida

Chem. Commun. 2024, 60, 4545.

[Selected as ChemComm HOT Articles]

https://doi.org/10.1039/D3CC05703H

126

Multisubstituted naphthalene synthesis from 4-hydroxy-2-pyrones and o-silylaryl triflates

K. Numata, S. Tabata, A. Kobayashi, *S. Yoshida

New J. Chem. 2023, 96, 401

https://doi.org/10.1039/D3NJ03831A

124

Synthesis of 1,2,3-triazoles using Grignard reactions through the protection of azides

R. Namioka, M. Suzuki, *S. Yoshida

Front. Chem. 2023, 11, 1237878.

https://doi.org/10.3389/fchem.2023.1237878

125

Facile synthesis of sulfinate esters from aryl iodides via direct oxidation of thioesters

K. Nakamura, Y. Kumagai, A. Kobayashi, M. Suzuki,

*S. Yoshida

Org. Biomol. Chem. 2023, 21, 6886.

https://doi.org/10.1039/D3OB01108A