Acylalkylation of Arynes Generated from o-Iodoaryl Triflates with Hydrosilanes and Cesium Fluoride

109

M. Minoshima, K. Uchida, Y. Nakamura, T. Hosoya,

*S. Yoshida

Diverse diaryl sulfide synthesis through consecutive aryne reactions

107

H. Nakajima, Y. Hazama, Y. Sakata, K. Uchida, T. Hosoya, *S. Yoshida

Chem. Commun. 2021, 57, 2621.

https://doi.org/10.1039/D0CC08373A

S1PR3–G12-biased agonist ALESIA targets cancer metabolism and promotes glucose starvation

108

M. Toyomoto, A. Inoue, K. Iida, M. Denawa, I. Kii, F. Marie, N. Kadji, T. Kishi, D. Im, T. Shimamura, H. Onogi, S. Yoshida, S. Iwata, J. Aoki, T. Hosoya, *M. Hagiwara

Cell Chem. Biol. 2021, in press.

https://doi.org/10.1016/j.chembiol.2021.01.004

Assembly of four modules onto a tetraazide platform by consecutive 1,2,3-triazole formations

106

*S. Yoshida, Y. Sakata, Y. Misawa, T. Morita, T. Kuribara, H. Ito, Y. Koike, I. Kii, *T. Hosoya

Chem. Commun. 2021, 57, 899.

https://doi.org/10.1039/D0CC07789E

Facile Synthesis of Tetraarylpyrazines by Sequential Cross-coupling Approach

105

Y. Nishiyama, K. Akiyama, Y. Sakata, T. Hosoya, *S. Yoshida

Chem. Lett. 2021, 50, 180.

https://doi.org/10.1246/cl.200715

Selected as Editor’s choice; Open Access

2-Azidoacrylamides as compact platforms for efficient modular synthesis

104

H. Takemura, S. Goto, T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 15541.

https://doi.org/10.1039/D0CC07212E

Single C−F Transformations of o‑Hydrosilyl Benzotrifluorides with Trityl Compounds as All-in-One Reagents

103

R. Idogawa, Y. Kim, K. Shimomori, T. Hosoya,

*S. Yoshida

Triazole formation of phosphinyl alkynes with azides through transient protection of phosphine by copper

102

N. Terashima, Y. Sakata, T. Meguro, T. Hosoya,

*S. Yoshida

Chem. Commun. 2020, 56, 14003.

https://doi.org/10.1039/D0CC06551J

Synthesis of Functionalized Benzopyran/Coumarin-Derived Aryne Precursors and Their Applications

101

Y. Nakamura, Y. Sakata, T. Hosoya, *S. Yoshida

One-step synthesis of benzo[b]thiophenes by aryne reaction with alkynyl sulfides

100

T. Matsuzawa, T. Hosoya, *S. Yoshida

Chem. Sci. 2020, 11, 9691.

https://doi.org/10.1039/D0SC04450D

Open Access; 化学工業日報; Highlighted in Chemistry Views

(Hexafluoroacetylacetonato)copper(I)–cycloalkyne complexes as protected cycloalkynes

99

N. Makio, T. Kuribara, K. Adachi, Y. Hatakeyama,

T. Meguro, Y. Sakata, K. Igawa, K. Tomooka, T. Hosoya,

*S. Yoshida

Chem. Commun. 2020, 56, 11449.

https://doi.org/10.1039/D0CC05182A

Open Access

Selective strain-promoted azide–alkyne cycloadditions through transient protection of bicyclo[6.1.0]nonynes with silver or gold

98

K. Adachi, T. Meguro, Y. Sakata, K. Igawa, K. Tomooka,

T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 9823.

https://doi.org/10.1039/D0CC04606J

Open Access

Synthesis of multisubstituted cycloalkenes through carbomagnesiation of strained cycloalkynes

97

Y. Tamura, Y. Minami, Y. Nishiyama, Y. Sakata, F. Karaki,

T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 7147.

https://doi.org/10.1039/D0CC02788J

Open Access

One-pot Synthesis of Allyl Sulfides from Sulfinate Esters and Allylsilanes through Reduction of Alkoxysulfonium Intermediates

96

A. Kobayashi, T. Matsuzawa, T. Hosoya, *S. Yoshida

Chem. Lett. 2020, 49, 813.

https://doi.org/10.1246/cl.200285

Open Access

Aryne Reaction and Cross-Coupling Approach for the Synthesis of Diverse N-Arylphenylalanine Derivatives

95

T. Kobayashi, T. Hosoya, *S. Yoshida

Chem. Lett. 2020, 49, 809.

https://doi.org/10.1246/cl.200276

Open Access

Synthesis of Diverse Aromatic Ketones through C–F Cleavage of Trifluoromethyl Group

94

M. Ikeda, T. Matsuzawa, T. Morita, T. Hosoya,

*S. Yoshida

Chem. Eur. J. 2020, 26, 12333.

https://doi.org/10.1002/chem.202001816

Synthesis of benzyl sulfides via substitution reaction at the sulfur of phosphinic acid thioesters

93

Y. Nishiyama, T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 5771.

https://doi.org/10.1039/D0CC02039G

Open Access

Sulfoxide Synthesis from Sulfinate Esters under Pummerer-like Conditions

92

A. Kobayashi, T. Matsuzawa, T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 5429.

https://doi.org/10.1039/D0CC02253E

Open Access

Synthesis of Thioxanthones through Formal C–H Thiolation of Benzoic Acid Esters and Acid-mediated Direct Cyclization

91

K. Mutsuura, Y. Sakata, K. Uchida, T. Hosoya,

*S. Yoshida

Chem. Lett. 2020, 49, 753

https://doi.org/10.1246/cl.200190

Open Access

A novel yellow fluorescent protein of recombinant apoPholasin with dehydrocoelenterazine

89

S. Inouye, Y. Miura-Sahara, R. Iimori, Y. Sakata,

Y. Hazama, S. Yoshida, M. Nakamura, T. Hosoya

Biochem. Biophys. Res. Commun. 2020, 526, 404.

https://doi.org/10.1016/j.bbrc.2020.03.085

Functionalization of a Single C–F Bond of Trifluoromethylarenes Assisted by an ortho-Silyl Group Using a Trityl-Based All-in-One Reagent with Ytterbium Triflate Catalyst

88

Y. Kim, K. Kanemoto, K. Shimomori, T. Hosoya,

*S. Yoshida

Chem. Eur. J. 2020, 26, 6136.

https://doi.org/10.1002/chem.202001315

Synthesis of Phenoxathiins and Phenothiazines by Aryne Reactions with Thiosulfonates

87

K. Kanemoto, Y. Sakata, T. Hosoya, *S. Yoshida

Chem. Lett. 2020, 49, 593.

https://doi.org/10.1246/cl.200132

Open Access

Facile assembly of three cycloalkyne-modules onto a platform compound bearing thiophene S,S-dioxide moiety and two azido groups

90

T. Meguro, Y. Sakata, T. Morita, T. Hosoya, *S. Yoshida

Chem. Commun. 2020, 56, 4720.

https://doi.org/10.1039/D0CC01810D

Open Access

Consecutive Aryne Generation Strategy for the Synthesis of 1,3-Diarylpyrazoles

86

T. Kobayashi, T. Hosoya, *S. Yoshida

J. Org. Chem. 2020, 85, 4448.

https://doi.org/10.1021/acs.joc.0c00172

HaloTag-based conjugation of proteins to barcoding-oligonucleotides

85

*J. Yazaki, Y. Kawashima, T. Ogawa, A. Kobayashi

M. Okoshi, T. Watanabe, S. Yoshida, I. Kii, S. Egami,

M. Amagai, T. Hosoya, K. Shiroguchi, O. Ohara

Nucl. Acid. Res. 2020, 48, e8.

https://doi.org/10.1093/nar/gkz1086

Open Access

Transition-Metal-Free Synthesis of N-Arylphenothiazines through an N- and S-Arylation Sequence

110

T. Matsuzawa, T. Hosoya, *S. Yoshida

Publication

Palladium-Catalyzed Sulfinylation of Aryl- and Alkenylborons with Sulfinate Esters

111

M. Suzuki, K. Kanemoto, Y. Nakamura, T. Hosoya,

*S. Yoshida

112

Nucleophilic transformations of azido-containing carbonyl compounds via protection of azido group

T. Aimi, T. Meguro, A. Kobayashi, *T. Hosoya, *S. Yoshida

Chem. Commun. 2021, 57, 6062.

https://doi.org/10.1039/D1CC01143J

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原著論文 (2020以降 / 2019~2016 / 2015以前)/総説・著書など特許

113

Facile Synthetic Methods for Diverse N-Arylphenylalanine Derivatives via Transformations of Aryne Intermediates and Cross-Coupling Reactions

T. Kobayashi, T. Hosoya, *S. Yoshida

Bull. Chem. Soc. Jpn. 2021, 94, 1823.

https://doi.org/10.1246/bcsj.20210149

114

Thioxanthone Synthesis from Benzoic Acid Esters through Directed ortho-Lithiation

A. Kobayashi, T. Matsuzawa, T. Hosoya, *S. Yoshida

Chem. Lett. 2021, 50, 1624. [Selected as Editor's Choice (優秀論文)]

https://doi.org/10.1246/cl.210293

115

Synthesis of Azidoanilines by the Buchwald–Hartwig Amination

Y. Sakata, S. Yoshida, *T. Hosoya

J. Org. Chem. 2021, 86, 15674.

https://doi.org/10.1021/acs.joc.1c02251

116

Multicomponent click assembly through 2-azidoacrylamides

having a nucleophilic amino group


H. Takemura, G. Orimoto, A. Kobayashi, T. Hosoya,

S. Yoshida*

Org. Biomol. Chem. 2022, 20, 6007.

[New Talent 2022 themed issue]

https://doi.org/10.1039/D2OB00151A

117

Hydride reduction of o-(fluorosilyl)benzodifluorides for subsequent C–F transformations

R. Idogawa, A. Kobayashi, Y. Kim, K. Shimomori, T. Hosoya, S. Yoshida*

Chem. Commun. 2022, 58, 3521.

https://doi.org/10.1039/D1CC06761C

118

Synthesis of Multisubstituted Benzenes from Phenols via Multisubstituted Benzynes


A. Nagai, A. Kobayashi, Y. Sakata, Y. Minami,

K. Uchida, T. Hosoya, S. Yoshida*

Synthesis 2022, 54, 5017.

[Special topic: Aryne Chemistry in Synthesis]

https://doi.org/10.1055/a-1834-2927

120

Pyridazine Synthesis from 1,2,4,5-Tetrazines and Alkynes in 1,1,1,3,3,3-Hexafluoro-2-propanol through the Inverse Electron Demand Diels–Alder Reaction

C. Yamamoto, M. Suzuki, S. Yoshida*

Bull. Chem. Soc. Jpn. 2022, 95, 1741. [BCSJ award article]

https://doi.org/10.1246/bcsj.20220267

119

Azido-type-selective triazole formation by iridium-catalyzed cycloaddition with thioalkynes


K. Sugiyama, Y. Sakata, T. Niwa, S. Yoshida, *T. Hosoya

Chem. Commun. 2022, 58, 6235.

https://doi.org/10.1039/D2CC01739C

121

Synthesis of benzo[b]furans from alkynyl sulfoxides and phenols by the interrupted Pummerer reaction

A. Kobayashi, T. Matsuzawa, T. Hosoya, S. Yoshida*

RSC Adv. 2023, 13, 839.

https://doi.org/10.1039/D2RA07856B

122

Migrative Thioamination of Aryne Intermediates Generated from o-Iodoaryl Triflates

S. Tabata, M. Minoshima, A. Kobayashi, T. Hosoya, S. Yoshida*

Synlett 2023, in press.

https://doi.org/10.1055/s-00000083


123

Fluorenones and Xanthones through Intramolecular C–F Arylation.

S. Hamada, S. Yoshida*

Bull. Chem. Soc. Jpn. 2023, in press.

https://doi.org/10.1246/bcsj.20230042